Compile Data Set for Download or QSAR
maximum 50k data
Found 67 of affinity data for UniProtKB/TrEMBL: P30098
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50299468(2-(3,4-dichlorophenyl)-N-(4-fluoro-3-trifluorometh...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50299468(2-(3,4-dichlorophenyl)-N-(4-fluoro-3-trifluorometh...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50299469(4-[4-(acetylmethyl-amino)-piperidin-1-yl]-2-(3,4-d...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50299469(4-[4-(acetylmethyl-amino)-piperidin-1-yl]-2-(3,4-d...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81944(CAS_86933-75-7 | NKB | NSC_5311312 | neuromedin K)
Affinity DataKi:  3.54nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50299470(4-[4-(acetylmethyl-amino)-piperidin-1-yl]-N-(2-chl...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50299470(4-[4-(acetylmethyl-amino)-piperidin-1-yl]-N-(2-chl...)
Affinity DataKi:  11.9nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  26nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50290297(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  54.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  208nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  2.31E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | FK 224 | NSC_6437864)
Affinity DataKi:  3.56E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50030178((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataKi:  5.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50212987(CHEMBL2110370 | GR-159897)
Affinity DataKi:  2.00E+4nMAssay Description:Tested for inhibition of binding of [3H]senktide to Tachykinin receptor 3 in guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50097909(1-[3-(5-Fluoro-1H-indol-3-yl)-ethyl]-4-(methylsulf...)
Affinity DataKi:  3.98E+4nMAssay Description:Tested for inhibition of binding of [3H]senktide to Tachykinin receptor 3 in guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 3 from guinea pig cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50403793(CHEMBL2115415)
Affinity DataIC50:  0.720nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50090485(CHEMBL295615 | spiro[(2-hydroxy)indane-1,40-piperi...)
Affinity DataIC50:  2.70nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050641(CHEMBL45340 | PD-161182 | [(R)-2-(2,3-Difluoro-phe...)
Affinity DataIC50:  3.70nMAssay Description:Compound was tested for binding affinity towards Tachykinin receptor 3 binding sites in guinea pig cortical membranes using [125I][MePhe7]-NKB as rad...More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050641(CHEMBL45340 | PD-161182 | [(R)-2-(2,3-Difluoro-phe...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I]-[MePhe7]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I]-[MePhe7]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  9nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against binding of [125I]-[MePhe7]-NKB SP to tachykinin NK-3 receptor in guinea pig cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50403790(CHEMBL2114963)
Affinity DataIC50:  11nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125I]-[MePhe7]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050652(CHEMBL47146 | PD-160946 | [(R)-2-(2-Fluoro-phenyl)...)
Affinity DataIC50:  14nMAssay Description:Compound was tested for binding affinity towards Tachykinin receptor 3 binding sites in guinea pig cortical membranes using [125I]-[MePhe7]-Neurokini...More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050652(CHEMBL47146 | PD-160946 | [(R)-2-(2-Fluoro-phenyl)...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I]-[MePhe7]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50282774(CHEMBL295301 | {(S)-1-[(R)-1-(8-Carbamoyl-octylcar...)
Affinity DataIC50:  15nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50090487(CHEMBL298247 | spiro[(2-hydroxy)indane-1,40-piperi...)
Affinity DataIC50:  17nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataIC50:  21nMAssay Description:NK3 IC50 determined using [125I]-Bolton Hunter labeled eledoisin at NK3 receptors from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50050642(CHEMBL296014 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against Tachykinin receptor 3 in guinea pig cortical membranes labeled with [125 I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  22nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50071484(CHEMBL308148 | N-[(R)-4-(4-Acetylamino-4-phenyl-pi...)
Affinity DataIC50:  208nMAssay Description:NK3 IC50 determined using [125I]-Bolton Hunter labeled eledoisin at NK3 receptors from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50283257((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...)
Affinity DataIC50:  276nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [3H]-Senktide to Tachykinin receptor 3 in the guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataIC50:  320nMAssay Description:Ability to displace [3H]senktide succinyl-[Asp9MePhe8]-SP (6-13)} from Tachykinin receptor 3 of guinea pig cerebral cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50403791(CHEMBL2114965)
Affinity DataIC50:  520nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50283253((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...)
Affinity DataIC50:  533nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [3H]-Senktide to Tachykinin receptor 3 in the guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50403792(CHEMBL2115416)
Affinity DataIC50:  660nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  717nMAssay Description:Inhibitory activity against binding of [125I]-[MePhe7]-NKB SP to tachykinin NK-3 receptor in guinea pig cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
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